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2013
  • Photos updated.( Doctor Thesis Presentation)(13 Dec 2013)
  • Lecturer Daisuke Urabe received Thieme Chemistry Journal Award 2014.
    (3 Dec 2013)
  • Hidenori Todoroki (G4) received "The Best Oral Presentation Award" at the 3rd ACP Junior Symposium. Title: "Synthetic Study of 4-Hydroxyzinowol" (30 Nov 2013)
  • Photos updated.(Boat Tournament)(19 Nov 2013)
  • Professor Masayuki Inoue received Mukaiyama Award Year 2014.
    (2 Oct 2013)
  • Publication Lists updated:
    D. Kamimura, D. Urabe, M. Nagatomo, M. Inoue, "Et3B]Mediated Radical-Polar Crossover Reaction for Single-Step Coupling of O,Te-Acetal, ,-Unsaturated Ketones, and Aldehydes/Ketones," Org. Lett. 2013, in press.
    DOI:10.1021/ol402563v
    (27 Sep 2013)
  • Publication Lists updated:
    T. Ishiyama, D. Urabe, H. Fujisawa, M. Inoue, "Concise Synthesis of the Multiply Oxygenated ABC-Ring System of the Dihydro--agarofurans," Org. Lett. 2013, in press.
    DOI:10.1021/ol402038b
    (31 Aug 2013)
  • Photos updated.(BBQ, Celebration for Passing Exam)(31 Aug 2013)
  • Publication Lists updated:
    K. Okura, M. Inoue, "The Orientation of the Terminal tBu Group of Antillatoxin is Important for Potent Toxicity: Design, Synthesis and Biological Evaluation of Conformationally Restricted Analogues of Antillatoxin," Asian J. Org. Chem. 2013, in press.
    DOI:10.1002/ajoc.201300111
    K. Okura, S. Matsuoka, M. Inoue, "The bulky side chain of antillatoxin is important for potent toxicity: rational design of photoresponsive cytotoxins based on SAR studies," Chem. Commun. 2013, in press.
    DOI:10.1039/C3CC44066D
    (1 Aug 2013)
  • Photos updated.(Group Photo)(29 Jun 2013)
  • Publication Lists updated:
    K. Sakata, D. Urabe, M. Inoue, "Preparation and palladium-mediated cross-coupling of -benzoyloxyalkylzinc bromides," Tetrahedron. Lett. 2013, in press.
    DOI:10.1016/j.tetlet.2013.05.114
    (4 Jun 2013)
  • Publication Lists updated:
    T. Hoshikawa, M. Inoue, "Photoinduced Direct 4-Pyridination of C(sp3)-H Bonds," Chem. Sci. 2013, in press.
    DOI:10.1039/C3SC51080H
    (27 May 2013)
  • Photos updated.(Sports Festival in Kemigawa)(25 May 2013)
  • Publication Lists updated:
    Y. Amaoka, M. Nagatomo, M. Inoue, "Metal-Free Fluorination of C(sp3)-H Bonds Using a Catalytic N-Oxyl Radical," Org. Lett. 2013, in press.
    DOI:10.1021/ol4006757
    (20 Apr 2013)
  • Publication Lists updated:
    K. Mukai, D. Urabe, S. Kasuya, N. Aoki, M. Inoue, "A Convergent Total Synthesis of 19-Hydroxysarmentogenin," Angew. Chem. Int. Ed. 2013, in press.
    DOI:10.1002/anie.201302067
    T. Tabuchi, D. Urabe, M. Inoue, "Asymmetric synthesis of a highly functionalized bicyclo[3.2.2]nonene derivative," Beilstein J. Org. Chem. 2013, 9, 655-663.
    DOI:10.3762/bjoc.9.74
    T. Shiba, Y. Kido, K. Sakamoto, D. K. Inaoka, C. Tsuge, R. Tatsumi, G. Takahashi, E. O. Balogun, T. Nara, T. Aoki, T. Honma, A. Tanaka, M. Inoue, S. Matsuoka, H. Saimoto, A. L. Moore, S. Harada, K. Kita, "Structure of the Trypanosome Cyanide-insensitive Alternative Oxidase, a Promising Drug Target," Proc. Natl. Acad. Sci. U.S.A. 2013, in press.
    DOI:10.1073/pnas.1218386110
    (11 Apr 2013)
  • Publication Lists updated:
    K. Murai, S. Katoh, D. Urabe, M. Inoue, "A radical-based approach for the construction of the tetracyclic structure of resiniferatoxin," Chem. Sci. 2013, in press.
    DOI:10.1039/C3SC50329A
    T. Kuranaga, Y. Sesoko, K. Sakata, N. Maeda, A. Hayata, M. Inoue, "Total Synthesis and Complete Structural Assignment of Yakufamide A," J. Am. Chem. Soc. 2013, in press.
    DOI:10.1021/ja401457h
    (3 Apr 2013)
  • Publication Lists (Reviews and Accounts) updated:
    H. Itoh, M. Inoue, "Chemical Construction and Structural Permutation of Potent Cytotoxin Polytheonamide B: Discovery of Artificial Peptides with Distinct Functions," Acc. Chem. Res. 2013, in press.
    DOI:10.1021/ar300315p
    (15 Mar 2013)
  • Publication Lists updated:
    T. Hoshikawa, S. Yoshioka, S. Kamijo, M. Inoue, "Photoinduced Direct Cyanation of C(sp3)-H Bonds" Synthesis 2013, in press.
    DOI:10.1055/s-0032-1318325
    Y. Isobe, M. Arita, R. Iwamoto, D. Urabe, H. Todoroki, K. Masuda, M. Inoue and H. Arai, "Stereochemical assignment and anti-inflammatory properties of the omega-3 lipid mediator resolvin E3," J. Biochem. 2013, in press.
    DOI:10.1093/jb/mvs151
    (4 Mar 2013)
  • Publication Lists updated:
    D. Urabe, M. Nagatomo, K. Hagiwara, K. Masuda, M. Inoue, "Symmetry-Driven Synthesis of 9-Demethyl-10,15-dideoxyryanodol" Chem. Sci. 2013, in press.
    DOI:10.1039/C3SC00023K (21 Jan 2013)
2012
  • Publication Lists updated:
    H. Itoh, M. Inoue, "Structural Permutation of Potent Cytotoxin, Polytheonamide B: Discovery of Cytotoxic Peptide with Altered Activity" ACS Med. Chem. Lett. 2012, in press.
    DOI:10.1021/ml300264c
    Y. Amaoka, S. Kamijo, T. Hoshikawa, M. Inoue, "Radical Amination of C(sp3)-H Bonds Using N-Hydroxyphthalimide and Dialkyl Azodicarboxylate" J. Org. Chem. 2012, in press.
    DOI:10.1021/jo301840e
  • "Featured Articles" is updated. (5 Nov 2012)
  • Publication Lists updated:
    T. Hoshikawa, S. Kamijo, M. Inoue, "Photochemically Induced Radical Alkynylation of C(sp3)-H Bonds" Org. Biomol. Chem. 2012, in press.
    DOI:10.1039/C2OB26785C (23 Oct 2012)
  • Our paper (N. Shinohara, H. Itoh, S. Matsuoka, M. Inoue "Selective Modification of the N-Terminal Structure of Polytheonamide B Significantly Changes its Cytotoxicity and Activity as an Ion Channel" ChemMedChem 2012, 7, 1770-1773.) has been placed on the back cover of ChemMedChem.
    DOI:10.1002/cmdc.201290052i14 Feb 2012j
  • Photos updated.(Lab Trip) (1 Sep 2012)
  • Publication Lists updated:
    H. Itoh, S. Matsuoka, M. Kreir, M. Inoue, "Design, Synthesis and Functional Analysis of Dansylated Polytheonamide Mimic: An Artificial Peptide Ion Channel" J. Am. Chem. Soc. 2012, 14011-14018.
    DOI:10.1021/ja303831a (27 Aug 2012)
  • Publication Lists updated:
    M. Iwatsu, D. Urabe, H. Todoroki, K. Masuda, M. Inoue, "Selective Introduction of Four Contiguous Stereocenters on the B-Ring of 4-Hydroxyzinowol" Heterocycles 2012, in press.
    DOI:10.3987/COM-12-S(N)76 (25 Aug 2012)
  • Photos updated.(Sports Festival in Kemigawa) (25 Aug 2012)
  • Publication Lists updated:
    D. Urabe, H. Yamaguchi, A. Someya, M. Inoue, "Intermolecular Radical Reaction of O,Se-Acetals Generated via Seleno-Pummerer Rearrangement" Org. Lett. 2012, in press.
    DOI:10.1021/ol301482f
    (20 Jul 2012)
  • Publication Lists updated:
    S. Kamijo, S. Matsumura, M. Inoue, "Microwave-assisted atom transfer radical addition of polychlorinated compounds to olefins without addition of metal catalysts" Tetrahedron Lett. 2012, in press.
    DOI:10.1016/j.tetlet.2012.06.027
    S. Kamijo, S. Yokosaka, M. Inoue, "Carbocyanation of trisubstituted olefins via Cu-catalyzed atom transfer radical addition" Tetrahedron Lett. 2012, in press.
    DOI:10.1016/j.tetlet.2012.06.004
    (26 Jun 2012)
  • Hiroki Yamaguchi (former member, G2) received Student Presentation Award at the 132 th Annual Meeting of the Pharmaceutical Society of Japan. Title: "Application of -Alkoxy Bridgehead Radical for Coupling of Oxygenated Carbocycles" (28 Apr 2012)
  • Publication Lists updated:
    N. Shinohara, H. Itoh, S. Matsuoka, M. Inoue, "Selective Modification of the N-Terminal Structure of Polytheonamide B Significantly Changes its Cytotoxicity and Activity as an Ion Channel" ChemMedChem 2012, in press.
    DOI:10.1002/cmdc.201200142 (19 Apr 2012)
  • Group Members updated.
    (6 Apr 2012)
  • Dr. Nagatomo has been promoted to assistant professor.
    (1 Apr 2012)
  • Dr. Kamijo has moved to Faculty of Science, Yamaguchi University.
    (31 Mar 2012)
  • Publication Lists updated:
    S. Matsuoka, M. Murai, T. Yamazaki, M. Inoue, "Short polyglutamine peptide forms a high-affinity binding site for thioflavin-T at the N-terminus" Org. Biomol. Chem. 2012, in press.
    DOI:10.1039/C2OB07157F
    D. Urabe, H. Todoroki, K. Masuda, M. Inoue, "Total syntheses of four possible stereoisomers of resolvin E3" Tetrahedron 2012, 3210-3219.
    DOI:10.1016/j.tet.2012.02.045 (21 Mar 2012)
  • Publication Lists updated:
    S. Kamijo, S. Yokosaka, M. Inoue, "Attachment of Carbonyl Functionalities onto Olefins via Copper-Promoted Radical Reaction of Dichloromethylcyanides" Tetrahedron 2012, in press.
    DOI:10.1016/j.tet.2012.01.089
    M. Inoue, "Total synthesis and functional analysis of non-ribosomal peptides," Chem. Rec. 2011, 11, 284-294.
    DOI:10.1002/tcr.201100014 (16 Feb 2012)
  • Publication Lists updated:
    S. Matsuoka, J. Mao, and M. Inoue, "Effects of the phosphatidylglycerol head group on the binding of short dermcidin-derived peptides to the phospholipid membrane surface" Tetrahedron Lett. 2012, 1078-1081.
    DOI:10.1016/j.tetlet.2011.12.071
    (1 Feb 2012)
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